Chemicals | Effects | Dosages | Solvent | ||
---|---|---|---|---|---|
LLC-PK cells | Caco-2 cells | MA104 cells | |||
Chlorpromazine | Inhibits clathrin-mediated endocytosis | 1 μM, 10 μM, 20 μM | 1 μM, 10 μM, 20 μM | 1 μM, 10 μM, 20 μM | DW |
Methyl-ß-cyclodextrin | Depletes cholesterol | 1 mM, 10 mM, 20 mM | 0.5 mM, 1 mM, 5 mM | 1 mM, 5 mM, 10 mM | DW |
Soluble cholesterol | Replenish cholesterol | 10 μM, 100 μM, 200 μM | 10 μM, 50 μM, 100 μM | 10 μM, 50 μM, 100 μM | DW |
Nystatin | Inhibits caveolae-mediated endocytosis, sequesters cholesterol | 1 μM, 10 μM, 25 μM | 1 μM, 10 μM, 25 μM | 1 μM, 25 μM, 50 μM | DMSO |
Dynasore | Inhibits dynamin | 1 μM, 50 μM, 100 μM | 1 μM, 50 μM, 100 μM | 1 μM, 50 μM, 100 μM | DMSO |
Chloroquine | Inhibits acidification of endosomes | 1 μM, 50 μM, 100 μM | – | – | DW |
Cytochalasin D | Disrupts actin cytoskeleton | 0.5 μM, 1 μM, 5 μM | – | – | DMSO |
Nocodazole | Disrupts microtubules | 1 μM, 10 μM, 20 μM | – | – | DMSO |
Amiloride | Inhibits macropinocytosis | 1 μM, 50 μM, 100 μM | – | – | DMSO |